SCHEMBL30684282

SCHEMBL30684282

Nc1cccc2c1ccn2-c1cn[nH]c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 5/20 0.34
HTR3A P46098 4/20 0.34
MAPT P10636 3/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
MAP4K4 O95819 1/20 0.33
CHEK1 O14757 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
CYP3A4 P08684 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30376189 0.80 HTR3A (0.44) HTR3AMAP4K4CHEK1ALDH1A1
SCHEMBL26698247 0.76 MAPT (0.37) ROCK1MAPTCYP3A4ALDH1A1LMNA
Hydrochloric Acid SCHEMBL30557207 0.73 BIRC5 (0.49) ROCK1HTR3AMAPTMAP4K4
SCHEMBL4880774 0.72 ALDH1A1 (0.44) ROCK1MAPTCYP3A4ALDH1A1HPGD
SCHEMBL4878604 0.72 MAPT (0.46) ROCK1MAPTMKNK1MKNK2CYP3A4
SCHEMBL15910764 0.72 SYK (0.41) HTR3AMAPTDDB1CRBN
Hydrochloric Acid SCHEMBL30376227 0.70 AKT1 (0.34) HTR3AMAPTMAP4K4CHEK1ALDH1A1
SCHEMBL3300423 0.69 RPS6KA5 (0.53) ROCK1MAPTMKNK1MKNK2CYP3A4
SCHEMBL29961184 0.69 RPS6KA5 (0.53) ROCK1MAPTMKNK1MKNK2CYP3A4
SCHEMBL30557228 0.66 CYP19A1 (0.58) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023235809-A1 CGAS INHIBITORS ELI LILLY AND COMPANY (US) 2023-12-07 WO disclosed