SCHEMBL30685709

SCHEMBL30685709

CCOC(=O)c1nn2c(c1C(F)(F)F)C(=O)NCC2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
ADORA1 P30542 3/20 0.35
MAPT P10636 3/20 0.34
KMT2A Q03164 2/20 0.34
PLAT P00750 1/20 0.34
ALDH1A1 P00352 2/20 0.34
CMA1 P23946 1/20 0.33
APP P05067 1/20 0.33
TSHR P16473 1/20 0.33
POLB P06746 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
KDM4E B2RXH2 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HPGD P15428 1/20 0.32
MEN1 O00255 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9940798 0.84 PARP1 (0.38) PARP1MAPTKMT2AALDH1A1TSHR
SCHEMBL9977655 0.81 PARP1 (0.37) PARP1ADORA1MAPTKMT2AALDH1A1
SCHEMBL26134476 0.81 PARP1 (0.37) PARP1MAPTKMT2AALDH1A1TSHR
SCHEMBL26135724 0.81 MAPT (0.37) PARP1MAPTKMT2AALDH1A1TSHR
SCHEMBL9938811 0.81 KDM5B (0.39) PARP1MAPTKMT2AALDH1A1APP
SCHEMBL26134848 0.80 PARP1 (0.36) PARP1MAPTKMT2AALDH1A1TSHR
SCHEMBL26134986 0.79 ELANE (0.35) PARP1PLATALDH1A1TSHRPOLB
SCHEMBL21130895 0.76 PDE4D (0.41) PARP1MAPTPLATALDH1A1TSHR
SCHEMBL26686728 0.75 KDM5B (0.38) PARP1MAPTKMT2AALDH1A1APP
SCHEMBL16699032 0.74 ADORA3 (0.37) PARP1KMT2APLATALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117279917-A Piperazine derivatives and their use in medicine 成都百裕制药股份有限公司 2023-12-22 CN disclosed