SCHEMBL30690356

SCHEMBL30690356

CC(=O)c1cc(C)cc2c(=O)n(C)c(-c3ccncc3)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP3A4 P08684 1/20 0.36
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP46A1 Q9Y6A2 1/20 0.36
GLA P06280 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
LMNA P02545 1/20 0.35
RECQL P46063 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GABRA1 P14867 2/20 0.34
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29139169 1.00 HTT (0.37) HTTCYP2C9CYP3A4KMT2AMEN1
SCHEMBL25359682 0.89 DHODH (0.45) KDM4EALDH1A1MAPTTDP1DHODH
SCHEMBL30690313 0.89 DHODH (0.45) KDM4EALDH1A1MAPTTDP1DHODH
SCHEMBL30495146 0.86 DHODH (0.38) KMT2AMEN1SMN1; SMN2NPSR1GABRA2
SCHEMBL25359989 0.86 DHODH (0.38) KMT2AMEN1SMN1; SMN2NPSR1GABRA2
SCHEMBL25358297 0.86 CYP2C9 (0.42) HTTCYP2C9CYP3A4KMT2AMEN1
SCHEMBL30495073 0.86 CYP2C9 (0.42) HTTCYP2C9CYP3A4KMT2AMEN1
SCHEMBL25360675 0.85 DHODH (0.32) CYP2C9KMT2AMEN1KDM4EALDH1A1
SCHEMBL30494959 0.85 DHODH (0.32) CYP2C9KMT2AMEN1KDM4EALDH1A1
SCHEMBL25360103 0.83 PTGS2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024026424-A1 QUINAZOLINONE DERIVATIVES AS AND RELATED USES BLACK DIAMOND THERAPEUTICS, INC. (US) 2024-02-01 WO disclosed
CN-117362281-A PI3K inhibitor and preparation method and application thereof 海创药业股份有限公司 2024-01-09 CN disclosed