SCHEMBL30706261

SCHEMBL30706261

NC(=O)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.55
PDPK1 O15530 1/20 0.55
TGM2 P21980 5/20 0.53
CES1 P23141 4/20 0.53
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA9 Q16790 1/20 0.53
MAOA P21397 5/20 0.49
MAOB P27338 5/20 0.49
ALDH1A1 P00352 1/20 0.49
CAPN9 O14815 1/20 0.47
CASP3 P42574 1/20 0.47
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5893915 1.00 SMYD3 (0.55) SMYD3PDPK1TGM2CES1CA12
SCHEMBL1050601 0.84 SMYD3 (0.56) SMYD3PDPK1TGM2CES1CA12
SCHEMBL29631093 0.84 SMYD3 (0.56) SMYD3PDPK1TGM2CES1CA12
SCHEMBL14563297 0.82 TGM2 (0.58) SMYD3TGM2CES1CA12CA1
SCHEMBL22380701 0.78 PDPK1 (0.57) SMYD3PDPK1TGM2CES1CA12
Acetamide SCHEMBL27380996 0.77 ROS1 (0.56) PDPK1TGM2CES1CA12CA1
SCHEMBL1290836 0.77 ACVR1 (0.62) PDPK1MAOAMAOBALDH1A1
SCHEMBL5783842 0.77 TGM2 (0.65) SMYD3TGM2CES1CA12CA1
SCHEMBL21154678 0.77 ACVR1 (0.62) PDPK1MAOAMAOBALDH1A1
SCHEMBL2360398 0.76 PPOX (0.48) PDPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115636817-B Isatin derivative containing triazole ring, and preparation method and application thereof 山东大学 2023-11-24 CN claimed