SCHEMBL30711990

SCHEMBL30711990

COC(=O)c1nn(C(F)F)c2cc(OCc3ccccc3)ccc12

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.51
F2 P00734 1/20 0.42
PLAU P00749 1/20 0.42
ELANE P08246 1/20 0.42
SRD5A2 P31213 1/20 0.42
S1PR3 Q99500 1/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 2/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAOB P27338 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CMKLR1 Q99788 1/20 0.41
DYRK1A Q13627 1/20 0.41
ROCK2 O75116 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19127310 1.00 HTR3A (0.51) HTR3AF2PLAUELANESRD5A2
SCHEMBL20646888 0.89 HTR3A (0.50) HTR3ASRD5A2S1PR3SMN1; SMN2MAOB
SCHEMBL20646891 0.87 HTR3A (0.49) HTR3ASRD5A2S1PR3LMNAMAOB
SCHEMBL23093693 0.83 ELANE (0.49) HTR3AF2PLAUELANEHPGD
SCHEMBL19128141 0.81 HTR3A (0.47) HTR3ASRD5A2MEN1KMT2ADYRK1A
SCHEMBL19128003 0.79 HTR3A (0.45) HTR3AF2PLAUELANESRD5A2
SCHEMBL19127270 0.79 ELANE (0.42) HTR3AF2PLAUELANEHPGD
SCHEMBL30711997 0.79 ELANE (0.42) HTR3AF2PLAUELANEHPGD
SCHEMBL28568174 0.78 ELANE (0.58) HTR3AF2PLAUELANEMEN1
SCHEMBL19128146 0.77 ELANE (0.42) F2PLAUELANESMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110869363-B 5-membered and bicyclic heterocyclic amides as ROCK inhibitors 百时美施贵宝公司 2024-01-05 CN disclosed