SCHEMBL30719409

SCHEMBL30719409

O=c1[nH]ccnc1-c1cncnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
TTK P33981 1/20 0.40
AURKB Q96GD4 1/20 0.40
INCENP Q9NQS7 1/20 0.40
KDM5B Q9UGL1 2/20 0.33
MAPT P10636 1/20 0.33
CYP2A6 P11509 1/20 0.32
GSK3B P49841 1/20 0.32
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MTOR P42345 1/20 0.31
ADK P55263 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
MAPK1 P28482 1/20 0.30
PIM1 P11309 1/20 0.30
ATM Q13315 1/20 0.30
PDE10A Q9Y233 1/20 0.30
KDM4A O75164 1/20 0.30
KDM4B O94953 1/20 0.30
KDM5C P41229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5065569 0.74 MTOR (0.53) MAPTALDH1A1MTORADKNISCH
SCHEMBL30719412 0.74 ACVR1 (0.41) AURKAAURKBINCENPKDM5BALDH1A1
SCHEMBL29096364 0.72 P2RX7 (0.37) KDM5BNISCHPIM1KDM4AKDM4B
SCHEMBL29948010 0.72 PDE3B (0.47) ALDH1A1NISCHMAPK1
SCHEMBL13619043 0.72 PDE3B (0.47) ALDH1A1SMN1; SMN2
SCHEMBL17151506 0.72 PDE3B (0.47)
SCHEMBL5065601 0.72 PDE3B (0.47) AURKAAURKBINCENPKDM5BMAPT
SCHEMBL13619228 0.72 NISCH (0.56) AURKBINCENPMAPTALDH1A1SMN1; SMN2
SCHEMBL1578108 0.71 NISCH (0.54) CYP2A6ALDH1A1SMN1; SMN2MTORADK
SCHEMBL14859149 0.70 AURKA (0.47) AURKATTKAURKBINCENPKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513020-B KDM1A inhibitors for the treatment of diseases 伊美格生物科学公司 2024-02-23 CN disclosed