SCHEMBL30723748

SCHEMBL30723748

COc1cc(Cl)ccc1C1=C(Br)CCCc2c1ccc1c2c(F)nn1C1CCCCO1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
DRD4 P21917 1/20 0.32
CRHR1 P34998 1/20 0.31
F11 P03951 3/20 0.31
KLKB1 P03952 3/20 0.31
CNR1 P21554 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTR2C P28335 3/20 0.31
SLC6A4 P31645 3/20 0.31
DGAT2 Q96PD7 1/20 0.31
EHMT2 Q96KQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30723867 0.88 NPC1 (0.33) NPC1RAB9ADRD4F11KLKB1
SCHEMBL30723941 0.87 NPC1 (0.34) NPC1RAB9ACRHR1F11KLKB1
SCHEMBL30723779 0.84 NPC1 (0.33) NPC1RAB9AF11KLKB1ALDH1A1
SCHEMBL30723843 0.76
SCHEMBL30723926 0.74 EHMT2 (0.32) EHMT2
SCHEMBL30723890 0.74 ESR1 (0.36)
SCHEMBL30723920 0.74
SCHEMBL30723815 0.73
SCHEMBL30723912 0.73
SCHEMBL25917542 0.72 CYP4F2 (0.34) ALDH1A1DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024006776-A1 ESTROGEN RECEPTOR ALPHA DEGRADERS AND MEDICAL USE THEREOF RELAY THERAPEUTICS, INC. (US) 2024-01-04 WO disclosed