SCHEMBL30725877

SCHEMBL30725877

O=C(Nc1ccc2[nH]nc(-c3cccnc3)c2c1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK7 P50613 1/20 0.67
JAK2 O60674 1/20 0.65
JAK1 P23458 1/20 0.65
AURKA O14965 1/20 0.64
CLK2 P49760 3/20 0.64
CLK3 P49761 3/20 0.64
DYRK1A Q13627 3/20 0.64
ITK Q08881 3/20 0.63
LRRK2 Q5S007 5/20 0.61
KCNK3 O14649 1/20 0.56
NTRK1 P04629 1/20 0.55
F2 P00734 1/20 0.55
F12 P00748 1/20 0.55
NAMPT P43490 2/20 0.54
IDO1 P14902 1/20 0.54
MAP2K4 P45985 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29172495 1.00 CDK7 (0.67) CDK7JAK2JAK1AURKACLK2
SCHEMBL8251866 0.90 JAK2 (0.74) CDK7JAK2JAK1AURKAITK
SCHEMBL30725858 0.90 DYRK1A (0.61) CDK7JAK2JAK1AURKACLK2
SCHEMBL29172497 0.90 LRRK2 (0.58) CDK7JAK2JAK1AURKACLK2
SCHEMBL29172502 0.90 DYRK1A (0.61) CDK7JAK2JAK1AURKACLK2
SCHEMBL30725869 0.90 LRRK2 (0.58) CDK7JAK2JAK1AURKACLK2
SCHEMBL29172484 0.88 PDPK1 (0.64) CDK7JAK2JAK1AURKACLK2
SCHEMBL30725844 0.88 PDPK1 (0.64) CDK7JAK2JAK1AURKACLK2
SCHEMBL30725862 0.88 PIM1 (0.60) CDK7JAK2JAK1AURKACLK2
SCHEMBL29172527 0.88 PIM1 (0.60) CDK7JAK2JAK1AURKACLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186066-A Indazole ALK5 inhibitor and preparation method and application thereof 中国药科大学 2023-12-08 CN disclosed