SCHEMBL30725858

SCHEMBL30725858

O=C(Nc1ccc2[nH]nc(-c3cccnc3)c2c1)c1ccc(F)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.61
CLK1 P49759 1/20 0.61
LRRK2 Q5S007 3/20 0.58
CYP11B1 P15538 2/20 0.57
CYP11B2 P19099 2/20 0.57
CDK7 P50613 1/20 0.55
ABL1 P00519 2/20 0.54
BCR P11274 2/20 0.54
PDGFRB P09619 1/20 0.54
PDGFRA P16234 1/20 0.54
NTRK1 P04629 2/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
CLK2 P49760 2/20 0.54
CLK3 P49761 2/20 0.54
AURKA O14965 1/20 0.53
JAK2 O60674 1/20 0.52
JAK1 P23458 1/20 0.52
WNT1 P04628 2/20 0.52
ITK Q08881 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29172502 1.00 DYRK1A (0.61) DYRK1ACLK1LRRK2CYP11B1CYP11B2
SCHEMBL30725877 0.90 CDK7 (0.67) DYRK1ALRRK2CDK7NTRK1CLK2
SCHEMBL29172495 0.90 CDK7 (0.67) DYRK1ALRRK2CDK7NTRK1CLK2
SCHEMBL29172484 0.89 PDPK1 (0.64) DYRK1ALRRK2CDK7NTRK1NPC1
SCHEMBL30725844 0.89 PDPK1 (0.64) DYRK1ALRRK2CDK7NTRK1NPC1
SCHEMBL5394136 0.89 LRRK2 (0.57) DYRK1ACLK1LRRK2CYP11B1CYP11B2
SCHEMBL29172497 0.89 LRRK2 (0.58) DYRK1ALRRK2CDK7CLK2CLK3
SCHEMBL30725869 0.89 LRRK2 (0.58) DYRK1ALRRK2CDK7CLK2CLK3
SCHEMBL5381989 0.87 AURKA (0.60) LRRK2NPC1RAB9AAURKAJAK2
SCHEMBL30725866 0.86 LRRK2 (0.70) LRRK2CYP11B1CYP11B2ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186066-A Indazole ALK5 inhibitor and preparation method and application thereof 中国药科大学 2023-12-08 CN disclosed