SCHEMBL30725869

SCHEMBL30725869

NC(=O)c1ccc(C(=O)Nc2ccc3[nH]nc(-c4cccnc4)c3c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.58
CDK7 P50613 1/20 0.55
JAK2 O60674 1/20 0.55
JAK1 P23458 1/20 0.55
CLK2 P49760 4/20 0.54
CLK3 P49761 4/20 0.54
DYRK1A Q13627 4/20 0.54
PIM1 P11309 2/20 0.53
AURKA O14965 1/20 0.53
MAP2K4 P45985 3/20 0.53
ITK Q08881 1/20 0.52
LMNA P02545 1/20 0.52
POLB P06746 1/20 0.52
MAPT P10636 1/20 0.52
MAPK1 P28482 1/20 0.50
MAPKAPK2 P49137 1/20 0.50
MAPKAPK3 Q16644 1/20 0.50
MAPK6 Q16659 1/20 0.50
MAPKAPK5 Q8IW41 1/20 0.50
ATR Q13535 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29172497 1.00 LRRK2 (0.58) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL30725862 0.92 PIM1 (0.60) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL29172527 0.92 PIM1 (0.60) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL30725877 0.90 CDK7 (0.67) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL29172495 0.90 CDK7 (0.67) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL29172502 0.89 DYRK1A (0.61) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL30725858 0.89 DYRK1A (0.61) LRRK2CDK7JAK2JAK1CLK2
SCHEMBL30725866 0.86 LRRK2 (0.70) LRRK2ITK
SCHEMBL29172510 0.86 LRRK2 (0.70) LRRK2ITK
SCHEMBL5373102 0.84 PIM1 (0.59) CDK7JAK2JAK1CLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186066-A Indazole ALK5 inhibitor and preparation method and application thereof 中国药科大学 2023-12-08 CN disclosed