SCHEMBL30728864

SCHEMBL30728864

COc1cccc(-c2cc(CBr)ccc2OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.56
HDAC4 P56524 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
CYP1A1 P04798 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2E1 P05181 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C8 P10632 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2A6 P11509 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP4B1 P13584 1/20 0.49
CYP2B6 P20813 1/20 0.49
CYP3A5 P20815 1/20 0.49
CYP2A7 P20853 1/20 0.49
CYP3A7 P24462 1/20 0.49
CYP2F1 P24903 1/20 0.49
CYP2C18 P33260 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14165291 0.88 CYP1A1 (0.61) PDE4BCYP1A1CYP1A2CYP2E1CYP3A4
SCHEMBL2936310 0.88 HDAC4 (0.56) PDE4BHDAC4HDAC2HDAC8CYP1A1
SCHEMBL10306550 0.86 PDE4B (0.57) PDE4BHDAC4HDAC2HDAC8CYP1A1
SCHEMBL15906086 0.85 SMN1; SMN2 (0.45) PDE4BHTR7MEN1LMNAHPGD
SCHEMBL29143285 0.84 HTR7 (0.51) PDE4BMAOBHTR7LMNAHPGD
SCHEMBL3466479 0.84 PDE4B (0.60) PDE4BHTR7TSHRALOX5GABRA1
SCHEMBL13578434 0.83 HTR7 (0.46) PDE4BHDAC4HDAC2HDAC8HTR7
SCHEMBL4936949 0.80 MAOB (0.54) HDAC4HDAC8CYP1A1CYP1A2CYP2E1
SCHEMBL8014205 0.80 PDE4B (0.46) PDE4BHDAC4HDAC2HDAC8CYP4F2
SCHEMBL3798654 0.80 PTPN5 (0.49) PDE4BMAOBLMNAHPGDCASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186001-B AHA1 inhibitor with multiple myeloma-resisting activity and preparation method and application thereof 南京中医药大学 2024-09-17 CN disclosed
CN-117186001-A AHA1 inhibitor with multiple myeloma-resisting activity and preparation method and application thereof 南京中医药大学 2023-12-08 CN disclosed