SCHEMBL30730783

SCHEMBL30730783

COc1cc(-c2cncc(-c3ccc(N4CCCC4=O)cc3)c2)c2cn[nH]c2n1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 2/20 0.43
HTT P42858 2/20 0.43
CYP11B1 P15538 3/20 0.39
CYP11B2 P19099 3/20 0.39
MAPT P10636 1/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
CHEK1 O14757 1/20 0.38
DGAT2 Q96PD7 1/20 0.37
PIP4K2A P48426 1/20 0.37
CD38 P28907 1/20 0.37
ATM Q13315 1/20 0.36
TNIK Q9UKE5 3/20 0.36
SYK P43405 1/20 0.35
TGFBR1 P36897 1/20 0.35
GRK6 P43250 1/20 0.35
HIF1A Q16665 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22554127 1.00 SMN1; SMN2 (0.43) SMN1; SMN2NPC1HTTCYP11B1CYP11B2
SCHEMBL22553760 0.86 PRKAB2 (0.40) NPC1CYP11B1CYP11B2CCNCCDK8
SCHEMBL30730822 0.86 PRKAB2 (0.40) NPC1CYP11B1CYP11B2CCNCCDK8
SCHEMBL22554087 0.85 SMN1; SMN2 (0.41) SMN1; SMN2NPC1HTTCYP11B1CYP11B2
SCHEMBL22554078 0.84 NPC1 (0.39) NPC1CCNCCDK8CD38TNIK
SCHEMBL30730823 0.84 NPC1 (0.39) NPC1CCNCCDK8CD38TNIK
SCHEMBL22553955 0.82 PIM1 (0.42) NPC1CYP11B2CCNCCDK8DGAT2
SCHEMBL22553920 0.80 TNIK (0.40) SMN1; SMN2NPC1CYP11B1CYP11B2CCNC
SCHEMBL22553792 0.80 SMN1; SMN2 (0.41) SMN1; SMN2NPC1HTTCYP11B1CYP11B2
SCHEMBL30730803 0.80 SMN1; SMN2 (0.41) SMN1; SMN2NPC1HTTCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed