SCHEMBL30730803

SCHEMBL30730803

COc1ncc(-c2cncc(-c3ccc(N4CCCC4=O)cc3)c2)c2cn[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 2/20 0.41
HTT P42858 1/20 0.41
CYP11B2 P19099 4/20 0.39
CYP11B1 P15538 3/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
CHEK1 O14757 1/20 0.38
DGAT2 Q96PD7 1/20 0.37
MAPT P10636 1/20 0.37
PIP4K2A P48426 1/20 0.37
PIM1 P11309 1/20 0.37
CD38 P28907 1/20 0.37
METAP2 P50579 2/20 0.36
CNR2 P34972 1/20 0.36
TGFBR1 P36897 1/20 0.35
GAA P10253 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22553792 1.00 SMN1; SMN2 (0.41) SMN1; SMN2NPC1HTTCYP11B2CYP11B1
SCHEMBL30730804 0.87 SMN1; SMN2 (0.42) SMN1; SMN2NPC1HTTCHEK1MAPT
SCHEMBL22553865 0.87 SMN1; SMN2 (0.42) SMN1; SMN2NPC1HTTCHEK1MAPT
SCHEMBL22553970 0.83 CYP11B1 (0.41) SMN1; SMN2NPC1HTTCYP11B2CYP11B1
SCHEMBL30730860 0.82 PIP4K2A (0.46) SMN1; SMN2NPC1HTTCYP11B2CYP11B1
SCHEMBL22553963 0.82 PIP4K2A (0.46) SMN1; SMN2NPC1HTTCYP11B2CYP11B1
SCHEMBL22554295 0.82 BRD4 (0.48) NPC1CCNCCDK8CHEK1PIP4K2A
SCHEMBL22554254 0.81 PRKAB2 (0.41) NPC1CYP11B2CYP11B1CCNCCDK8
SCHEMBL22553817 0.81 CYP11B2 (0.41) SMN1; SMN2NPC1HTTCYP11B2CYP11B1
SCHEMBL30730784 0.81 CYP11B2 (0.41) SMN1; SMN2NPC1HTTCYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed