SCHEMBL30734178

SCHEMBL30734178

Nc1cc(-c2ccc3ncnc(N4CCN(c5ccc(F)cc5)CC4)c3n2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 10/20 0.49
MINK1 Q8N4C8 1/20 0.49
TNIK Q9UKE5 1/20 0.49
ACHE P22303 1/20 0.45
BACE1 P56817 1/20 0.45
PIM1 P11309 1/20 0.44
PIM3 Q86V86 1/20 0.44
PIM2 Q9P1W9 1/20 0.44
MAPT P10636 3/20 0.43
HTT P42858 1/20 0.43
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
THRB P10828 1/20 0.41
MKNK1 Q9BUB5 2/20 0.41
MKNK2 Q9HBH9 2/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30734142 0.89 MAP4K4 (0.44) MAP4K4MINK1TNIKPIM1PIM3
SCHEMBL30734141 0.89 MAP4K4 (0.46) MAP4K4MINK1TNIKACHEBACE1
SCHEMBL30734199 0.83 MAP4K4 (0.47) MAP4K4MINK1TNIKMAPTHTT
SCHEMBL30734233 0.83 ACHE (0.55) MAP4K4ACHEBACE1MAPTHTT
SCHEMBL30734219 0.81 ACHE (0.47) MAP4K4MINK1TNIKACHEBACE1
SCHEMBL30734209 0.78 MAP4K4 (0.47) MAP4K4MINK1TNIKMAPTHTT
SCHEMBL30734202 0.77 MAP4K4 (0.43) MAP4K4MINK1TNIKMKNK1MKNK2
SCHEMBL31745185 0.75 PIM1 (0.44) MAP4K4MINK1TNIKPIM1PIM3
SCHEMBL4526207 0.75 MKNK1 (0.55) MAP4K4MAPTHTTLMNATP53
SCHEMBL30734154 0.74 MAPT (0.51) ACHEBACE1MAPTHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250382301-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF UNIV ARIZONA (US) 2025-12-18 US disclosed
EP-4543888-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF Arizona Board of Regents on behalf of The University of Arizona (US) 2025-04-30 EP disclosed
WO-2023250083-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2023-12-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250382301-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF CLK2, CLK3, CLK1 MAP4K4 107/4885MINK1 118/4885TNIK 380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.