SCHEMBL30734200

SCHEMBL30734200

Brc1ccc2ncnc(N3CCC4(CCN(c5ccccn5)C4)CC3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.54
ALDH1A1 P00352 12/20 0.51
NPSR1 Q6W5P4 1/20 0.51
ACHE P22303 1/20 0.50
BACE1 P56817 1/20 0.50
HSD17B10 Q99714 11/20 0.46
HPGD P15428 9/20 0.46
CYP3A4 P08684 7/20 0.46
TSHR P16473 7/20 0.45
CYP2D6 P10635 6/20 0.45
CYP2C19 P33261 5/20 0.45
CYP1A2 P05177 5/20 0.45
CYP2C9 P11712 5/20 0.45
USP2 O75604 3/20 0.45
PDGFRB P09619 1/20 0.44
MAPK1 P28482 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30734183 0.96 HTT (0.51) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30734194 0.87 HTT (0.66) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30734214 0.84 HTT (0.62) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30734144 0.82 ACHE (0.45) ALDH1A1ACHEBACE1HSD17B10HPGD
SCHEMBL30734177 0.80 HTT (0.69) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30902257 0.78 HTT (0.63) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30333781 0.78 HTT (0.70) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30734149 0.78 HTT (0.47) HTTALDH1A1NPSR1ACHEBACE1
SCHEMBL30734174 0.78 ACHE (0.45) ALDH1A1ACHEBACE1HSD17B10HPGD
SCHEMBL30734135 0.76 HTT (0.71) HTTALDH1A1NPSR1ACHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4543888-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF Arizona Board of Regents on behalf of The University of Arizona (US) 2025-04-30 EP disclosed
WO-2023250083-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2023-12-28 WO disclosed