SCHEMBL30737254

SCHEMBL30737254

COCCn1cc(-c2cccc(O)c2)nn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.51
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50
CD74 P04233 3/20 0.49
MIF P14174 3/20 0.49
HDAC8 Q9BY41 8/20 0.47
HDAC6 Q9UBN7 8/20 0.47
HDAC3 O15379 7/20 0.47
HDAC4 P56524 7/20 0.47
HDAC1 Q13547 7/20 0.47
HDAC7 Q8WUI4 7/20 0.47
HDAC2 Q92769 7/20 0.47
HDAC10 Q969S8 7/20 0.47
HDAC11 Q96DB2 7/20 0.47
HDAC9 Q9UKV0 7/20 0.47
HDAC5 Q9UQL6 7/20 0.47
SRC P12931 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GPR55 Q9Y2T6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28311174 0.84 TEK (0.55) ALOX5CD74MIFHDAC8HDAC6
SCHEMBL30737470 0.82 ALOX5 (0.57) ALOX5HSD17B1HSD17B2CD74MIF
SCHEMBL18760619 0.81 ALOX5 (0.56) ALOX5HSD17B1HSD17B2CD74MIF
SCHEMBL19690458 0.80 HDAC8 (0.54) ALOX5HSD17B1HSD17B2HDAC8HDAC6
SCHEMBL30737267 0.77 HDAC3 (0.48) ALOX5HSD17B1HSD17B2CD74MIF
SCHEMBL28875514 0.76 HDAC3 (0.44) CD74MIFHDAC8HDAC6HDAC3
SCHEMBL16271204 0.75 MEN1 (0.54) HDAC8HDAC6HDAC3HDAC4HDAC1
SCHEMBL12986809 0.75 ALOX5 (0.56) ALOX5HSD17B1HSD17B2CD74MIF
SCHEMBL13172900 0.74 SRC (0.52) ALOX5HSD17B1HSD17B2CD74MIF
SCHEMBL30737158 0.74 HDAC3 (0.45) ALOX5HSD17B1HSD17B2CD74MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4543858-A1 BIFUNCTIONAL MOLECULES THAT SELECTIVELY INDUCE DEGRADATION OF EXTRACELLULAR TARGETS IN LYSOSOMES Draupnir Bio ApS (DK) 2025-04-30 EP disclosed
WO-2023247754-A1 BIFUNCTIONAL MOLECULES THAT SELECTIVELY INDUCE DEGRADATION OF EXTRACELLULAR TARGETS IN LYSOSOMES DRAUPNIR BIO APS (DK) 2023-12-28 WO disclosed