SCHEMBL30737553

SCHEMBL30737553

N#CCC(=O)c1ccc(C(=O)N2CC3(CC(=O)C3)C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
GPR183 P32249 7/20 0.38
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.35
AR P10275 3/20 0.34
CYP3A4 P08684 2/20 0.33
ALDH1A1 P00352 2/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30737566 0.81 CECR2 (0.41) GAAGPR183TSHRMEN1LMNA
SCHEMBL30737654 0.76 HPGD (0.56) TSHRMEN1LMNAKMT2AALDH1A1
SCHEMBL30737599 0.76 HPGD (0.61) TSHRMEN1LMNAKMT2AALDH1A1
SCHEMBL30737498 0.75 HPGD (0.65) TSHRMEN1LMNAKMT2AALDH1A1
SCHEMBL30737764 0.73 ACACB (0.47) GPR183TSHRCYP3A4ALDH1A1HPGD
SCHEMBL395103 0.73 GSK3B (0.48) GAAMEN1KMT2ACYP3A4ALDH1A1
SCHEMBL11770219 0.66 CYP19A1 (0.57) GAALMNAALDH1A1PKMHPGD
SCHEMBL14918493 0.66 TSHR (0.52) TSHRALDH1A1
SCHEMBL1568921 0.65 GSK3B (0.57) GAALMNAALDH1A1HPGD
SCHEMBL3659298 0.65 TPMT (0.46) GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117510505-A Pyrimidopyrazoles derivatives and their use in medicine 中国药科大学 2024-02-06 CN disclosed