SCHEMBL30739017

SCHEMBL30739017

COc1ccc2c(=O)n(Br)c(CCl)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.47
CYP3A4 P08684 5/20 0.46
ALDH1A1 P00352 3/20 0.42
GFER P55789 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
KMT2A Q03164 2/20 0.41
USP2 O75604 1/20 0.41
GLA P06280 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
KCNH2 Q12809 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
CYP1A2 P05177 2/20 0.40
MEN1 O00255 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
GABRA1 P14867 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1161537 0.85 CYP3A4 (0.55) PDE10ACYP3A4ALDH1A1GFERSMN1; SMN2
SCHEMBL1161533 0.74 CYP3A4 (0.55) PDE10ACYP3A4ALDH1A1SMN1; SMN2KMT2A
SCHEMBL1663473 0.71 LMNA (0.63) PDE10ACYP3A4ALDH1A1SMN1; SMN2KMT2A
SCHEMBL1464928 0.70 CYP3A4 (0.56) PDE10ACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL31267402 0.70 ALDH1A1 (0.55) ALDH1A1GFERSMN1; SMN2MAPTRAB9A
SCHEMBL30186041 0.69 KDM4E (0.59) ALDH1A1KMT2AMAPTRAB9AMEN1
SCHEMBL6930235 0.69 KDM4E (0.59) ALDH1A1KMT2AMAPTRAB9AMEN1
SCHEMBL4394401 0.69 USP2 (0.77) CYP3A4ALDH1A1SMN1; SMN2KMT2AUSP2
SCHEMBL28694003 0.69 SMN1; SMN2 (0.65) PDE10ACYP3A4SMN1; SMN2KMT2AUSP2
SCHEMBL29260843 0.69 SMN1; SMN2 (0.49) PDE10ACYP3A4ALDH1A1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117561258-A Novel substituted tricyclic aza heterocycles as SOS1 inhibitors 唯久生物技术(苏州)有限公司 2024-02-13 CN disclosed