SCHEMBL30745018

SCHEMBL30745018

CCOC(=O)c1nc2ccc(O)cc2cc1OC(C)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
CA12 O43570 4/20 0.43
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA7 P43166 4/20 0.43
CA9 Q16790 4/20 0.43
CA14 Q9ULX7 4/20 0.43
TSHR P16473 1/20 0.42
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 2/20 0.41
MIF P14174 1/20 0.41
PFKFB3 Q16875 1/20 0.41
HPGD P15428 1/20 0.41
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
MEN1 O00255 1/20 0.39
HSP90AA1 P07900 1/20 0.39
KMT2A Q03164 1/20 0.39
GLP1R P43220 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745012 0.81 MEN1 (0.66) MAOBALDH1A1HPGDMEN1HSP90AA1
SCHEMBL30744965 0.76 CA12 (0.43) MAOAMAOBCA12CA1CA2
SCHEMBL20944030 0.76 ALDH1A1 (0.51) MAOAMAOBCA12CA1CA2
SCHEMBL13313476 0.75 S1PR4 (0.45) TSHRKDM4EALDH1A1MEN1KMT2A
SCHEMBL14089785 0.74 TSHR (0.72) MAOAMAOBCA12CA1CA2
SCHEMBL2004474 0.73 ESR1 (0.49) CA12CA1CA2CA7CA9
SCHEMBL2210778 0.72 CYP1A2 (0.54) MAOAMAOBCA12CA1CA2
SCHEMBL5430440 0.72 CYP1A2 (0.46) TSHRKDM4EALDH1A1MEN1KMT2A
SCHEMBL6643041 0.72 KDM4E (0.47) MAOBCA12CA2CA7CA9
SCHEMBL21865495 0.70 CA12 (0.48) MAOAMAOBCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111295382-B Bridged bicyclic compounds as farnesyl ester X receptor modulators 百时美施贵宝公司 2024-02-02 CN disclosed