SCHEMBL30745170

SCHEMBL30745170

COc1cccc(CNC=O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
ALDH1A1 P00352 4/20 0.56
HTT P42858 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MMP13 P45452 1/20 0.55
HDAC1 Q13547 2/20 0.54
ADH1B P00325 1/20 0.53
ADH1C P00326 1/20 0.53
ADH1A P07327 1/20 0.53
ADH7 P40394 1/20 0.53
KDM4E B2RXH2 2/20 0.52
HPGD P15428 2/20 0.52
USP2 O75604 1/20 0.52
HDAC3 O15379 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
CHRM1 P11229 2/20 0.51
CHRM3 P20309 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3305893 1.00 CHRM2 (0.59) CHRM2MEN1KMT2AALDH1A1HTT
SCHEMBL3305905 0.94 ALDH1A1 (0.57) CHRM2MEN1KMT2AALDH1A1HTT
SCHEMBL24061767 0.94 CHRM2 (0.54) CHRM2MEN1KMT2AALDH1A1HTT
SCHEMBL24061766 0.89 ALDH1A1 (0.68) CHRM2MEN1KMT2AALDH1A1HTT
SCHEMBL1134127 0.83 CHRM2 (0.74) CHRM2MEN1KMT2AALDH1A1HTT
SCHEMBL5548185 0.83 SMN1; SMN2 (0.57) CHRM2ALDH1A1SMN1; SMN2ADH1BADH1C
SCHEMBL2473241 0.83 CHRM2 (0.66) CHRM2MEN1KMT2AALDH1A1KDM4E
SCHEMBL22912213 0.83 ALDH1A1 (0.56) CHRM2MEN1KMT2AALDH1A1HTT
SCHEMBL5537789 0.82 ADH1B (0.49) MEN1KMT2AALDH1A1HTTSMN1; SMN2
SCHEMBL4881807 0.82 TSHR (0.51) MEN1KMT2AALDH1A1SMN1; SMN2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113956249-B Brain-targeted AChE inhibitor prodrug, and preparation method and application thereof 中国药科大学 2024-02-02 CN claimed
CN-113956249-B Brain-targeted AChE inhibitor prodrug, and preparation method and application thereof 中国药科大学 2024-02-02 CN disclosed