SCHEMBL30757446

SCHEMBL30757446

CCCCC(=O)Nc1c(C#N)cnn1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.43
PTGS1 P23219 3/20 0.42
PTGS2 P35354 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 2/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK10 P53779 1/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20540355 0.78 SMN1; SMN2 (0.54) TSHRSMN1; SMN2ALDH1A1TP53HPGD
SCHEMBL10617379 0.77 PTGS1 (0.47) TSHRSMN1; SMN2ALDH1A1HPGDPTGS1
SCHEMBL8997373 0.74 POLB (0.39) SMN1; SMN2ALDH1A1TP53HPGDCYP1A2
SCHEMBL12629794 0.74 RAB9A (0.51) SMN1; SMN2RAB9AMEN1KMT2AMAPK10
SCHEMBL11094611 0.74 PTGS1 (0.42) TSHRSMN1; SMN2ALDH1A1PTGS1PTGS2
SCHEMBL10618486 0.74 PTGS1 (0.46) TSHRSMN1; SMN2HPGDPTGS1PTGS2
SCHEMBL10617044 0.73 PTGS1 (0.46) TSHRSMN1; SMN2PTGS1PTGS2RAB9A
SCHEMBL10618027 0.73 PTGS1 (0.46) TSHRSMN1; SMN2PTGS1PTGS2RAB9A
SCHEMBL8997213 0.72 GFER (0.64) TSHRALDH1A1PTGS1PTGS2GFER
SCHEMBL8997219 0.71 PTGS1 (0.58) TSHRSMN1; SMN2ALDH1A1TP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023224963-A1 DUAL-ACTING ANGIOTENSIN AND ENDOTHELIN RECEPTOR ANTAGONISTS ARIA PHARMACEUTICALS, INC. (US) 2023-11-23 WO disclosed