SCHEMBL30760140

SCHEMBL30760140

Cc1nccnc1-c1ccc([C@H](CO)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 1/20 0.39
AAK1 Q2M2I8 2/20 0.38
CYP17A1 P05093 2/20 0.37
RIPK1 Q13546 1/20 0.36
PTPRB P23467 3/20 0.36
ROCK2 O75116 3/20 0.36
ROCK1 Q13464 3/20 0.36
MAPK13 O15264 1/20 0.36
RPS6KA5 O75582 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
PRKCG P05129 1/20 0.36
CDK1 P06493 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CDK2 P24941 1/20 0.36
MAPK1 P28482 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
CLK2 P49760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30760064 0.85 MKNK1 (0.45) AAK1CYP17A1RIPK1PTPRBROCK2
SCHEMBL30760051 0.83 TRPV1 (0.45) AAK1RIPK1ROCK2ROCK1MAPK13
SCHEMBL30760154 0.82 ROCK2 (0.43) AAK1CYP17A1RIPK1PTPRBROCK2
SCHEMBL30760073 0.81 HDAC4 (0.40) AAK1CYP17A1PTPRBROCK2ROCK1
SCHEMBL28995700 0.80 PPARG (0.45) RIPK1MEN1ALDH1A1LMNAHPGD
SCHEMBL17619268 0.80 PPARG (0.45) RIPK1MEN1ALDH1A1LMNAHPGD
SCHEMBL19580931 0.80 VHL (0.46) PTPRB
SCHEMBL30759976 0.80 HDAC4 (0.45) AAK1CYP17A1RIPK1PTPRBROCK2
SCHEMBL18551023 0.80 VHL (0.46) PTPRB
SCHEMBL14831426 0.79 CTSK (0.52) RIPK1ROCK2ROCK1MAPK13RPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024040080-A1 KRAS INHIBITOR CONJUGATES ERASCA, INC. (US) 2024-02-22 WO disclosed