SCHEMBL30761102

SCHEMBL30761102

O=C(Nc1ccc(F)cn1)c1cc(Cl)c(F)cn1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.53
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
CYP3A4 P08684 4/20 0.48
FFAR2 O15552 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
ALDH1A1 P00352 1/20 0.48
PKM P14618 1/20 0.48
TSHR P16473 1/20 0.48
CYP1A2 P05177 3/20 0.47
CYP2C9 P11712 3/20 0.47
KCNH2 Q12809 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
BRD4 O60885 1/20 0.47
SLC6A3 Q01959 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3852931 0.77 NPC1 (0.60) GRM5NPC1RAB9ACYP3A4FFAR2
SCHEMBL4187822 0.76 GRM5 (0.51) GRM5NPC1RAB9ACYP3A4FFAR2
SCHEMBL30761114 0.76 GRM5 (0.49) GRM5CYP3A4CYP1A2CYP2C9KCNH2
SCHEMBL31224325 0.75 NPC1 (0.42) NPC1RAB9ACYP3A4SMN1; SMN2ALDH1A1
SCHEMBL4858178 0.75 F10 (0.57) GRM5NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL30761121 0.75 DYRK1A (0.46) GRM5
SCHEMBL30761214 0.75 NPC1 (0.59) GRM5NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL7904776 0.74 GRM5 (0.72) GRM5CYP3A4CYP1A2CYP2C9KCNH2
SCHEMBL18145934 0.74 NPC1 (0.53) GRM5NPC1RAB9ACYP3A4FFAR2
SCHEMBL18160436 0.74 RAB9A (0.67) GRM5NPC1RAB9AFFAR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059204-A1 HETEROARYL ANALOGS AS MGLU5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSITY (US) 2024-03-21 WO disclosed