SCHEMBL30772995

SCHEMBL30772995

C#Cc1ccc2cnccc2n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.37
MELK Q14680 1/20 0.34
GRM5 P41594 1/20 0.33
KCNH2 Q12809 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
MALT1 Q9UDY8 1/20 0.32
IMPDH2 P12268 2/20 0.32
ROCK2 O75116 1/20 0.31
CTSA P10619 1/20 0.31
HTT P42858 2/20 0.31
PRKCZ Q05513 1/20 0.31
MIF P14174 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
NCOA1 Q15788 1/20 0.30
NCOA3 Q9Y6Q9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27856307 0.84 MAP4K4 (0.39) HDAC8MELKGRM5KCNH2PRKCZ
SCHEMBL987561 0.80 NQO1 (0.47) MELKGRM5KCNH2HTTNCOA3
SCHEMBL2007578 0.80 PDE3B (0.36) MELKGRM5KCNH2PDE3BPDE3A
SCHEMBL740158 0.72 GRM5 (0.53) GRM5KCNH2MIFKDM4EALDH1A1
SCHEMBL30824468 0.72 GRM5 (0.53) GRM5KCNH2MIFKDM4EALDH1A1
SCHEMBL1899820 0.72 NPC1 (0.47) PDE3BPDE3AMALT1IMPDH2ROCK2
SCHEMBL208412 0.69
SCHEMBL276051 0.68 KDM4E (0.41) MELKPDE3BPDE3AMALT1IMPDH2
SCHEMBL3064494 0.68 IMPDH2 (0.42) KCNH2PDE3BPDE3AMALT1IMPDH2
SCHEMBL3952608 0.68 MALT1 (0.37) PDE3BPDE3AMALT1IMPDH2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117157292-A KRAS G12D inhibitors and uses thereof 苏州赞荣医药科技有限公司 2023-12-01 CN disclosed