SCHEMBL740158

SCHEMBL740158

C#Cc1ccc2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.53
KCNH2 Q12809 1/20 0.53
NCF1 P14598 3/20 0.46
CYP1A2 P05177 2/20 0.46
NOS2 P35228 1/20 0.46
BACE1 P56817 1/20 0.46
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
TTR P02766 1/20 0.45
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
GLA P06280 1/20 0.42
HPGD P15428 1/20 0.42
ACHE P22303 1/20 0.42
MGAM O43451 1/20 0.41
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
AR P10275 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30824468 1.00 GRM5 (0.53) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL15940575 0.94 GRM5 (0.49) GRM5KCNH2NCF1CYP1A2NOS2
Thiophene SCHEMBL15940611 0.89 GRM5 (0.45) GRM5KCNH2NCF1CYP1A2NOS2
Toluene SCHEMBL27946106 0.89 CYP1A2 (0.47) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL15940691 0.83 GRM5 (0.41) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL10788654 0.77 GRM5 (0.53) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL29359679 0.77 GRM5 (0.53) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL194312 0.77 GRM5 (0.53) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL3059086 0.77 GRM5 (0.53) GRM5KCNH2NCF1CYP1A2NOS2
SCHEMBL75226 0.77 GRM5 (0.53) GRM5KCNH2NCF1CYP1A2NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 103 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106083813-A A kind of synthetic method of triazole quinolines 太原理工大学 2016-11-09 CN claimed
CN-120442103-A Preparation method of cold-resistant low-temperature printing ink 哈尔滨金龙盛印刷材料有限公司 2025-08-08 CN disclosed
US-20250163088-A1 HALF-SANDWICH TRANSITION METAL COMPLEXES AND USES THEREOF DEBRECENI EGYETEM (HU) 2025-05-22 US disclosed
CN-119912441-A Novel oxazolidinone compound and anti-infection application thereof 安徽医科大学第一附属医院 2025-05-02 CN disclosed
CN-119792542-A Method for accelerating bio-orthogonal catalysis of acid/reduction sensitive polymer vesicles in situ of tumor 苏州大学 2025-04-11 CN disclosed
WO-2025076285-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USING THE SAME DELPHIA THERAPEUTICS, INC. (US) 2025-04-10 WO disclosed
EP-4463230-A1 HALF-SANDWICH TRANSITION METAL COMPLEXES AND USES THEREOF Debreceni Egyetem (HU) 2024-11-20 EP disclosed
WO-2024051720-A1 5-PYRIDINE-1H-INDAZOLE COMPOUND FOR TARGETED INHIBITION OF CLK2 AND USE OF COMPOUND 中国药科大学 2024-03-14 WO disclosed
CN-115304583-B 5-pyridine-1H-indazole compound for targeted inhibition of CLK2 and application thereof 中国药科大学 2023-07-21 CN disclosed
WO-2023041947-A1 HALF-SANDWICH TRANSITION METAL COMPLEXES AND USES THEREOF DEBRECENI EGYETEM (HU) 2023-03-23 WO disclosed
US-20050192212-A1 Macrocyclic peptides active against the hepatitis C virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-09-01 US disclosed
WO-2005070955-A1 MACROCYCLIC PEPTIDES ACTIVE AGAINST THE HEPATITIS C VIRUS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-08-04 WO disclosed
US-20050165052-A1 Substituted quinolines for the treatment of protozoa and retrovirus co-infections INSTITUT DE RECHERCHE POUR LE DEVELOPPEMENT (FR) 2005-07-28 US disclosed
CN-1200925-C Aromatic carboxylic acid compound, acid halide derivative thereof, and process for producing the same SUMITOMO BAKELITE CO (JP) 2005-05-11 CN disclosed
US-20040068139-A1 Aromatic carboxylic acids, acid halides thereof and processes for preparing both SUMITOMO BAKELITE COMPANY, LTD. (JP) 2004-04-08 US disclosed
CN-1474800-A Aromatic carboxylic acid compound, acid halide derivative thereof, and process for producing the same 住友电木株式会社 2004-02-11 CN disclosed
EP-1351940-A1 SUBSTITUTED QUINOLINES FOR THE TREATMENT OF PROTOZOAN AND RETROVIRUS CO-INFECTIONS Institut de Recherche pour le Développement ( IRD) (FR) 2003-10-15 EP disclosed
EP-1346975-A1 AROMATIC CARBOXYLIC ACIDS, ACID HALIDES THEREOF AND PROCESSES FOR PREPARING BOTH SUMITOMO BAKELITE CO., LTD. (JP) 2003-09-24 EP disclosed
WO-2002057238-A1 SUBSTITUTED QUINOLINES FOR THE TREATMENT OF PROTOZOAN AND RETROVIRUS CO-INFECTIONS INSTITUT DE RECHERCHE POUR LE DEVELOPPEMENT (IRD) (FR) 2002-07-25 WO disclosed
WO-2002055077-A1 USE OF IMIDAZOLYL CYCLIC ACETAL DERIVATIVES IN THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF DISEASES MEDIATED BY THE ALK5 RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2002-07-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050192212-A1 Macrocyclic peptides active against the hepatitis C virus CTRL, RNPEP, RNASE1 GRM5 4838/4885KCNH2 2609/4885NCF1 2188/4885
US-20050165052-A1 Substituted quinolines for the treatment of protozoa and retrovirus co-infections C1S, C5, NSFL1C GRM5 2484/4885KCNH2 259/4885NCF1 2296/4885
US-20040068139-A1 Aromatic carboxylic acids, acid halides thereof and processes for preparing both CCR1, CCRL2, CCR6 GRM5 3878/4885KCNH2 2712/4885NCF1 1540/4885
US-20250163088-A1 HALF-SANDWICH TRANSITION METAL COMPLEXES AND USES THEREOF SLC39A3, CUTA, SLC30A6 GRM5 3296/4885KCNH2 4631/4885NCF1 1508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.