SCHEMBL30777928

SCHEMBL30777928

COc1cc(F)ccc1-c1cc(Cl)ncc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 11/20 0.48
GSK3A P49840 1/20 0.48
IRAK1 P51617 1/20 0.48
CDK2 P24941 7/20 0.47
CCNT1 O60563 3/20 0.47
CCNK O75909 2/20 0.47
CDK1 P06493 2/20 0.47
CCNE1 P24864 1/20 0.47
CDK12 Q9NYV4 1/20 0.47
GPBAR1 Q8TDU6 2/20 0.46
HDAC3 O15379 4/20 0.44
HDAC1 Q13547 3/20 0.44
HDAC6 Q9UBN7 3/20 0.44
KCNQ3 O43525 1/20 0.42
KCNQ2 O43526 1/20 0.42
KCNH2 Q12809 2/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15649934 1.00 CDK9 (0.48) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL18416745 0.86 HSP90AA1 (0.46) KCNQ3KCNQ2
SCHEMBL15720877 0.85 KCNQ3 (0.42) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL12098360 0.83 GPBAR1 (0.43) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL12098356 0.82 GPBAR1 (0.43) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL30507433 0.82 CDK9 (0.54) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL15650695 0.82 CDK9 (0.54) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL15682390 0.77 F2RL1 (0.40) CDK9GSK3AIRAK1CDK2CCNT1
SCHEMBL14785028 0.77 CDK2 (0.50) CDK9CDK2CCNT1CCNE1
SCHEMBL29944149 0.77 CDK2 (0.50) CDK9CDK2CCNT1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683020-A Aminopyridine compound of phthalazinone, preparation method thereof and application thereof in preparation of inhibitor and antitumor drug 华南理工大学 2024-03-12 CN disclosed
CN-117510513-A Heterocyclic compounds having biological activity 首药控股(北京)股份有限公司 2024-02-06 CN disclosed