SCHEMBL307825

SCHEMBL307825

CC1(C)O[C@@H]2[C@H](O1)[C@@H](CO)O[C@H]2n1cnc2c(O)nc(O)nc21

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.65
PI4K2B Q8TCG2 1/20 0.65
PI4K2A Q9BTU6 1/20 0.65
PI4KB Q9UBF8 1/20 0.65
LMNA P02545 2/20 0.57
ALDH1A1 P00352 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
RXFP1 Q9HBX9 1/20 0.47
P2RX1 P51575 1/20 0.45
P2RX3 P56373 1/20 0.45
P2RX4 Q99571 1/20 0.45
TP53 P04637 1/20 0.42
CYP2C19 P33261 1/20 0.42
ADORA3 P0DMS8 3/20 0.41
ADORA1 P30542 3/20 0.41
ADORA2A P29274 2/20 0.41
GAA P10253 1/20 0.41
ADORA2B P29275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260752 0.89 PI4KA (0.69) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL260760 0.88 PI4KA (0.59) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL2291671 0.85 PI4KA (0.80) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL22757346 0.83 PI4KA (0.64) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL23914964 0.82 LMNA (0.65) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL18493278 0.82 LMNA (0.65) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL17205571 0.82 LMNA (0.65) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL24601301 0.82 PI4KA (0.55) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL24601294 0.82 PI4KA (0.55) PI4KAPI4K2BPI4K2API4KBLMNA
SCHEMBL24601293 0.82 PI4KA (0.55) PI4KAPI4K2BPI4K2API4KBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093380-B2 Viricides, antitumor agents, anticancer agents PHARMASSET, INC. (US) 2012-01-10 US disclosed
EP-1545545-A4 COMPOUNDS WITH THE BICYCLO 4.2.1 NONANE SYSTEM FOR THE TREATMENT OF i FLAVIVIRIDAE /i INFECTIONS PHARMASSET INC (US) 2008-09-03 EP disclosed
EP-1545545-A2 COMPOUNDS WITH THE BICYCLO 4.2.1 NONANE SYSTEM FOR THE TREATMENT OF i FLAVIVIRIDAE /i INFECTIONS Pharmasset, Inc. (US) 2005-06-29 EP disclosed
US-20040082574-A1 Compounds with the bicyclo[4.2.1]nonane system for the treatment of flavivridae infections PHARMASSET, INC. 2004-04-29 US disclosed
WO-2004013300-A2 COMPOUNDS WITH THE BICYCLO[4.2.1]NONANE SYSTEM FOR THE TREATMENT OF FLAVIVIRIDAE INFECTIONS PHARMASSET INC. (US) 2004-02-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082574-A1 Compounds with the bicyclo[4.2.1]nonane system for the treatment of flavivridae infections CYP4B1, HAVCR2, CYP2S1 PI4KA 187/4885PI4K2B 240/4885PI4K2A 191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.