SCHEMBL30792011

SCHEMBL30792011

COC(=O)c1ccc(CO[Si](C)(C)C(C)(C)C)nc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.50
KDM4E B2RXH2 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
MAPT P10636 3/20 0.41
GABRA5 P31644 6/20 0.40
ALDH1A1 P00352 2/20 0.40
RAB9A P51151 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8682205 1.00 MAPK1 (0.50) MAPK1KDM4EL3MBTL1CA12CA1
SCHEMBL15835801 0.88 MAPK1 (0.47) MAPK1KDM4EL3MBTL1MAPTGABRA5
SCHEMBL8545215 0.85 MAPT (0.46) L3MBTL1MAPTGABRA5ALDH1A1
SCHEMBL20483548 0.82 HDAC6 (0.38) L3MBTL1
SCHEMBL1439028 0.82 MAPK1 (0.59) MAPK1KDM4EL3MBTL1CA12CA1
SCHEMBL1313112 0.81 LOXL2 (0.51) MAPK1KDM4EL3MBTL1CA12CA1
SCHEMBL8681688 0.81 NPC1 (0.38) ALDH1A1RAB9AKMT2AGAANPC1
SCHEMBL30746942 0.80 MAPK1 (0.46) MAPK1KDM4EL3MBTL1CA1CA2
SCHEMBL9521091 0.80 GABRA5 (0.36) KDM4EL3MBTL1GABRA5ALDH1A1KMT2A
SCHEMBL507626 0.80 HRH3 (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114302886-B Triazolopyridazine derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2024-03-22 CN disclosed