SCHEMBL307962

SCHEMBL307962

COc1ccccc1N(C(=O)CC(N)=O)c1ccc(Oc2ccnc3cc(C(=O)NN(C)C)sc23)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.44
KDR P35968 19/20 0.44
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2C Q14957 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL895543 0.80 MET (0.41) METKDR
SCHEMBL306874 0.78 KDR (0.49) METKDRGRIN3BGRIN1GRIN2C
SCHEMBL18487310 0.78 MET (0.43) METKDR
SCHEMBL307961 0.77 MET (0.65) METKDR
SCHEMBL308564 0.77 KDR (0.46) METKDRGRIN3BGRIN1GRIN2C
SCHEMBL306717 0.76 MET (0.42) METKDR
SCHEMBL896589 0.75 MET (0.70) METKDR
SCHEMBL10272795 0.75 KDR (0.47) METKDR
SCHEMBL14230733 0.75 MET (0.70) METKDR
SCHEMBL306922 0.73 KDR (0.46) METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093264-B2 Fused heterocycles as inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE INC. (CA) 2012-01-10 US disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 MET 2/4885KDR 4/4885GRIN3B 1864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.