Hydroxyflutamide

Hydroxyflutamide

SCHEMBL3079778

CC(C)(O)C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 1.00
CYP3A4 P08684 2/20 1.00
PGR P06401 1/20 1.00
CES2 O00748 1/20 0.68
ABCB11 O95342 1/20 0.68
ALDH1A1 P00352 1/20 0.68
LMNA P02545 1/20 0.68
CYP1A2 P05177 1/20 0.68
GLA P06280 1/20 0.68
ADORA3 P0DMS8 1/20 0.68
CHRM1 P11229 1/20 0.68
CYP2C9 P11712 1/20 0.68
ALOX15 P16050 1/20 0.68
TSHR P16473 1/20 0.68
TBXA2R P21731 1/20 0.68
AADAC P22760 1/20 0.68
MAPK1 P28482 1/20 0.68
CYP2C19 P33261 1/20 0.68
ADRA1A P35348 1/20 0.68
HTT P42858 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydroxyflutamide SCHEMBL29379312 1.00 AR (1.00) ARCYP3A4PGRCES2ABCB11
Hydroxyflutamide SCHEMBL10395764 0.96 AR (0.93) ARCYP3A4PGRCES2ABCB11
Hydroxyflutamide SCHEMBL10395767 0.96 AR (0.93) ARCYP3A4PGRCES2ABCB11
SCHEMBL11407111 0.92 AR (0.85) ARCYP3A4PGRCES2ABCB11
SCHEMBL14086876 0.91 AR (0.83) ARCYP3A4PGRCES2ABCB11
SCHEMBL2011994 0.90 AR (0.82) ARCYP3A4PGRCES2ABCB11
SCHEMBL7524151 0.90 AR (0.81) ARCYP3A4PGRCES2ABCB11
SCHEMBL14086877 0.90 AR (0.81) ARCYP3A4PGRCES2ABCB11
SCHEMBL8409001 0.89 AR (0.81) ARCYP3A4PGRCES2ABCB11
SCHEMBL8410375 0.88 AR (0.79) ARCYP3A4PGRCES2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1738752-A1 Pharmaceutical combinations comprising cis-retine acid Schering Aktiengesellschaft (DE) 2007-01-03 EP claimed
EP-1641458-A2 PHARMACEUTICAL COMBINATIONS OF PHTHALAZINE VEGF INHIBITORS AND BENZAMIDE HDAC INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2006-04-05 EP claimed
US-20050054647-A1 New pharmaceutical combination BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2005-03-10 US claimed
WO-2004058234-A2 PHARMACEUTICAL COMBINATIONS OF PHTHALAZINE VEGF INHIBITORS AND BENZAMIDE HDAC INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2004-07-15 WO claimed
US-4598072-A Combinations of an aromatase-inhibitor and an antiandrogen for prophylaxis and/or treatment of benign prostatic hyperplasia SCHERING AKTIENGESELLSCHAFT (DE) 1986-07-01 US claimed
US-4039684-A 4-NITRO-3-TRIFLUOROMETHYL-ISOBUTYRANILIDE OR CORRESPONDING 2-HYDROXY- COMPOUND SCHERING CORPORATION (US) 1977-08-02 US claimed
WO-2024010817-A2 SELECTIVE ANDROGEN RECEPTOR DEGRADER (SARD) O-LINKED LIGANDS AND METHODS OF USE THEREOF UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2024-01-11 WO disclosed
US-20230382870-A1 N-AROMATIC AMIDE COMPOUNDS, PREPARATION METHODS AND USES THEREOF SHENZHEN EDK PHARMACEUTICAL TECH CO LTD (CN) 2023-11-30 US disclosed
EP-3357513-B1 PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF KANGPU BIOPHARMACEUTICALS LTD (CN) 2023-10-25 EP disclosed
EP-3357513-B1 PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF KANGPU BIOPHARMACEUTICALS LTD (CN) 2023-10-25 EP disclosed
US-11760727-B2 N-aromatic amide compounds, preparation methods and uses thereof SHENZHEN EDK PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2023-09-19 US disclosed
US-20230227492-A1 MONOMERIC AND OLIGOMERIC COMPOUND EMBODIMENTS AS CONTRACEPTIVES AND THERAPIES AND METHODS OF MAKING AND USING THE SAME THE USA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2023-07-20 US disclosed
EP-4164743-A2 MONOMERIC AND OLIGOMERIC COMPOUND EMBODIMENTS AS CONTRACEPTIVES AND THERAPIES AND METHODS OF MAKING AND USING THE SAME The United States of America, as represented by The Secretary, Department of Health and Human Services (US) 2023-04-19 EP disclosed
WO-1992016233-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF PROSTATIC CANCER CONTAINING A 5 ALPHA REDUCTASE INHIBITOR AND AN ANTIANDROGEN MERCK & CO., INC. (US) 1992-10-01 WO disclosed
US-4921941-A TRIPEPTIDE ESTERS SCHERING CORPORATION (US) 1990-05-01 US disclosed
EP-0348564-A1 Orally active antiandrogens SCHERING CORPORATION (US) 1990-01-03 EP disclosed
WO-1989000165-A1 ORALLY ACTIVE ANTIANDROGENS SCHERING CORPORATION (US) 1989-01-12 WO disclosed
US-4598072-A Combinations of an aromatase-inhibitor and an antiandrogen for prophylaxis and/or treatment of benign prostatic hyperplasia SCHERING AKTIENGESELLSCHAFT (DE) 1986-07-01 US disclosed
US-4039684-A 4-NITRO-3-TRIFLUOROMETHYL-ISOBUTYRANILIDE OR CORRESPONDING 2-HYDROXY- COMPOUND SCHERING CORPORATION (US) 1977-08-02 US disclosed
US-4039684-A 4-NITRO-3-TRIFLUOROMETHYL-ISOBUTYRANILIDE OR CORRESPONDING 2-HYDROXY- COMPOUND SCHERING CORPORATION (US) 1977-08-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227492-A1 MONOMERIC AND OLIGOMERIC COMPOUND EMBODIMENTS AS CONTRACEPTIVES AND THERAPIES AND METHODS OF MAKING AND USING THE SAME SHBG, CYP19A1, GNRHR AR 7/4885CYP3A4 2085/4885PGR 16/4885
US-20050054647-A1 New pharmaceutical combination VEGFA, INHA, PGF AR 300/4885CYP3A4 1151/4885PGR 116/4885
US-20230382870-A1 N-AROMATIC AMIDE COMPOUNDS, PREPARATION METHODS AND USES THEREOF H1-3, H1-0, NAT1 AR 385/4885CYP3A4 687/4885PGR 1068/4885
US-11760727-B2 N-aromatic amide compounds, preparation methods and uses thereof AR, BPHL, CYP19A1 AR 1/4885CYP3A4 239/4885PGR 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.