SCHEMBL30799052

SCHEMBL30799052

C#CCn1cc([N+](=O)[O-])c(=O)n(C)c1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 4/20 0.43
MAPT P10636 3/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GLA P06280 1/20 0.34
BLM P54132 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GAA P10253 1/20 0.31
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480361 0.73 MAPT (0.50) ADORA2BMAPTKDM4ELMNAHTT
SCHEMBL30799164 0.67 ADORA2B (0.43) ADORA2BMAPTKDM4ELMNAGLA
SCHEMBL10562805 0.62
SCHEMBL316763 0.61 ADORA2B (1.00) ADORA2BMAPTLMNAGLABLM
SCHEMBL9409708 0.60 ADORA2B (0.42) ADORA2BGLABLMADORA3KMT2A
SCHEMBL29620659 0.60 ALDH1A1 (0.34) MAPT
SCHEMBL11480035 0.59 KDM4E (0.50) ADORA2BMAPTKDM4ELMNAHTT
SCHEMBL2256402 0.59 MAPT (0.55) MAPTKDM4ELMNAHTTNPSR1
SCHEMBL29042327 0.59 MAPT (0.55) MAPTKDM4ELMNAHTTNPSR1
SCHEMBL15804011 0.59 MAPT (0.55) MAPTKDM4ELMNAHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024050825-A1 COMPOUNDS AS MLKL INHIBITORS NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2024-03-14 WO disclosed