SCHEMBL30814652

SCHEMBL30814652

O=C(N1CCc2c(Br)ccc(F)c2C1)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.45
ESR2 Q92731 4/20 0.45
ABHD6 Q9BV23 6/20 0.43
HTR5A P47898 5/20 0.38
EP300 Q09472 1/20 0.37
CREBBP Q92793 1/20 0.37
PKM P14618 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
RBP4 P02753 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17114724 0.94 ESR1 (0.45) ESR1ESR2ABHD6HTR5AEP300
SCHEMBL28901664 0.84 HTR5A (0.40) ABHD6HTR5APTGDR2
SCHEMBL19693487 0.83 ABHD6 (0.44) ESR1ESR2ABHD6EP300CREBBP
SCHEMBL17798326 0.80 ESR1 (0.45) ESR1ESR2ABHD6EP300CREBBP
SCHEMBL506312 0.79 ESR1 (0.43) ESR1ESR2ABHD6EP300CREBBP
SCHEMBL22981209 0.79 ESR1 (0.53) ESR1ESR2ABHD6PKM
SCHEMBL19643352 0.79 ESR1 (0.53) ESR1ESR2ABHD6HTR5AEP300
SCHEMBL17114829 0.79 ESR1 (0.44) ESR1ESR2ABHD6HTR5AEP300
SCHEMBL31163315 0.79 ESR2 (0.47) ESR2ABHD6
SCHEMBL587897 0.77 ABHD6 (0.69) ESR1ESR2ABHD6HTR5AEP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024046221-A1 EGFR INHIBITORS AND USES THEREOF DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2024-03-07 WO disclosed