SCHEMBL30817828

SCHEMBL30817828

O=C(NC1CCC(Oc2cc(N3CCOCC3)cc3ncncc23)CC1)C1COC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 5/20 0.38
LMNA P02545 2/20 0.38
GAA P10253 2/20 0.38
PIK3CD O00329 1/20 0.37
PIK3R1 P27986 1/20 0.37
ERBB2 P04626 3/20 0.37
CYP46A1 Q9Y6A2 1/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BMPR1B O00238 1/20 0.34
BMPR1A P36894 1/20 0.34
TGFBR1 P36897 1/20 0.34
ACVRL1 P37023 1/20 0.34
ACVR1 Q04771 1/20 0.34
SIK1 P57059 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177846 1.00 PRKDC (0.38) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL21177843 1.00 PRKDC (0.38) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL21177841 0.95 LMNA (0.41) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL21177861 0.95 LMNA (0.41) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL21177844 0.95 LMNA (0.41) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL21187288 0.95 LMNA (0.41) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL30823286 0.95 LMNA (0.41) PRKDCLMNAGAAPIK3CDPIK3R1
SCHEMBL21179454 0.89 ERBB2 (0.38) PRKDCERBB2BMPR1BBMPR1ATGFBR1
SCHEMBL21179453 0.89 ERBB2 (0.38) PRKDCERBB2BMPR1BBMPR1ATGFBR1
SCHEMBL21187304 0.87 ERBB2 (0.35) PRKDCLMNAGAAPIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111757876-B DNA-PK inhibitors 沃泰克斯药物股份有限公司 2024-03-22 CN disclosed
EP-3740480-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2024-03-06 EP disclosed