SCHEMBL30820

SCHEMBL30820

CC(=O)c1ccc(C(F)(F)F)cc1[AsH2]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.50
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 3/20 0.49
KDM4E B2RXH2 2/20 0.49
USP2 O75604 1/20 0.49
CYP2C19 P33261 1/20 0.49
CFTR P13569 1/20 0.46
MAPT P10636 2/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GAA P10253 1/20 0.42
SORT1 Q99523 2/20 0.41
RXFP1 Q9HBX9 2/20 0.40
ALOX15 P16050 1/20 0.40
NOTUM Q6P988 1/20 0.40
CES1 P23141 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
NR4A1 P22736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29499840 0.83 GAA (0.58) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL1350804 0.83 GAA (0.58) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL21852902 0.82 CES2 (0.55) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL18291815 0.81 ALDH1A1 (0.56) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL1451777 0.79 MAPT (0.57) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL1996550 0.79 CES2 (0.72) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL29540816 0.79 MAPT (0.57) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL30481870 0.79 CES2 (0.72) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL20810 0.78 ALDH1A1 (0.71) CES2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL2477164 0.78 CES2 (0.50) CES2ALDH1A1HPGDHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609085-A1 SUBSTITUTED QUINOLINE-3-CARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2013-07-03 EP disclosed
WO-2012025238-A1 SUBSTITUTED QUINOLINE-3-CARBOXAMIDES AS KCNQ2/3 MODULATORS Grünenthal GmbH (DE) 2012-03-01 WO disclosed