SCHEMBL30823709

SCHEMBL30823709

Cn1cnc(-c2ccccc2C(N)=O)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 6/20 0.49
HCRTR2 O43614 6/20 0.49
DPP4 P27487 1/20 0.46
BCAT2 O15382 1/20 0.46
CSNK1A1 P48729 1/20 0.44
TYRO3 Q06418 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
KDM4E B2RXH2 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
GRM5 P41594 1/20 0.41
NUDT1 P36639 1/20 0.40
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11079561 0.75 BCAT2 (0.46) DPP4BCAT2CSNK1A1TYRO3DYRK1B
SCHEMBL997870 0.74 CSNK1A1 (0.57) BCAT2CSNK1A1TYRO3DYRK1BKDM4E
SCHEMBL31227695 0.74 CSNK1A1 (0.57) BCAT2CSNK1A1TYRO3DYRK1BKDM4E
SCHEMBL30964842 0.74 BCAT2 (0.53) DPP4BCAT2CSNK1A1TYRO3DYRK1B
SCHEMBL1380693 0.74 BCAT2 (0.53) DPP4BCAT2CSNK1A1TYRO3DYRK1B
SCHEMBL30823708 0.74 HCRTR1 (0.41) HCRTR1HCRTR2MAPK1
SCHEMBL11908649 0.74 HCRTR2 (0.70) HCRTR1HCRTR2
SCHEMBL31280858 0.72 TYK2 (0.40) HCRTR1HCRTR2CSNK1A1DYRK1B
SCHEMBL210767 0.71 BCAT2 (0.74) BCAT2CSNK1A1TYRO3DYRK1BKDM4E
SCHEMBL30514077 0.71 BCAT2 (0.74) BCAT2CSNK1A1TYRO3DYRK1BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111655681-B Heterocyclylamino-substituted triazoles as modulators of Rho-related protein kinases 莱德克斯制药公共有限公司 2024-01-05 CN disclosed