SCHEMBL30829491

SCHEMBL30829491

COC(=O)c1c(I)c(C)nn1Cc1nc(-c2ccc(C(F)(F)F)cc2)c(C=CC(=O)OC(C)(C)C)s1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 15/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
ENPP2 Q13822 1/20 0.32
PPARA Q07869 4/20 0.32
PPARG P37231 2/20 0.32
FFAR1 O14842 1/20 0.32
DHODH Q02127 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
HSP90AA1 P07900 1/20 0.32
MAPT P10636 1/20 0.32
CRHBP P24387 1/20 0.32
KMT2A Q03164 1/20 0.32
CRHR2 Q13324 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29231402 0.93 PPARD (0.35) PPARDENPP2PPARAPPARGFFAR1
SCHEMBL21542468 0.86 CA12 (0.32) PPARDNPC1ALDH1A1GAAENPP2
SCHEMBL20214039 0.86 CA12 (0.32) PPARDNPC1ALDH1A1GAAENPP2
SCHEMBL28346707 0.79 PTGER1 (0.34) PPARDNPC1ALDH1A1GAAENPP2
SCHEMBL20214017 0.73 KDM4E (0.33) ALDH1A1GAADHODHKDM4EMEN1
SCHEMBL20213964 0.70 ALDH1A1 (0.34) PPARDNPC1ALDH1A1GAADHODH
SCHEMBL20213979 0.69 ALDH1A1 (0.38) PPARDNPC1ALDH1A1GAADHODH
SCHEMBL20214002 0.65 ALDH1A1 (0.35) PPARDNPC1ALDH1A1GAADHODH
SCHEMBL2362965 0.64 SCN9A (0.45) ALDH1A1GAAKDM4EMEN1MAPT
SCHEMBL29231533 0.63 XPO1 (0.39) DHODHPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110603254-B Substituted pyrazole compounds and methods of using the same for treating hyperproliferative diseases 班塔姆制药有限责任公司 2024-04-12 CN disclosed