SCHEMBL30831996

SCHEMBL30831996

CN(C(=O)NCC1CCN(CC(=O)c2ccc(F)cc2)CC1)c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
TSHR P16473 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HTT P42858 1/20 0.48
HTR2A P28223 5/20 0.45
HTR2C P28335 4/20 0.45
KCNH2 Q12809 1/20 0.45
HTR1A P08908 2/20 0.45
TMEM97 Q5BJF2 2/20 0.45
DRD2 P14416 3/20 0.43
SIGMAR1 Q99720 3/20 0.43
HTR2B P41595 2/20 0.43
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP3A4 P08684 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29207981 0.95 ALDH1A1 (0.44) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
SCHEMBL30832004 0.86 HTR2A (0.42) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
SCHEMBL30832015 0.85 HTR2A (0.52) ALDH1A1TSHRSMN1; SMN2HTR2AHTR2C
SCHEMBL30832041 0.84 MEN1 (0.42) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
Trifluoroacetic Acid SCHEMBL29208033 0.82 HTR2A (0.41) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
SCHEMBL29280894 0.81 MEN1 (0.55) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
SCHEMBL30840071 0.81 MEN1 (0.55) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
Trifluoroacetic Acid SCHEMBL29207974 0.81 HTR2A (0.48) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL30832006 0.79 KDM4E (0.47) ALDH1A1TSHRSMN1; SMN2KDM4EHTT
SCHEMBL29280915 0.76 HTR2A (0.61) KDM4EHTR2AHTR2CKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed