SCHEMBL30832004

SCHEMBL30832004

Cc1cccc(N(C)C(=O)NCC2CCN(CC(=O)c3ccc(F)cc3)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.42
HTR2C P28335 3/20 0.42
KCNH2 Q12809 1/20 0.42
HTR1A P08908 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
DRD2 P14416 2/20 0.42
HTR2B P41595 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
TSHR P16473 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
USP2 O75604 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29208033 0.95 HTR2A (0.41) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL30832041 0.88 MEN1 (0.42) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL30831996 0.86 ALDH1A1 (0.48) HTR2AHTR2CKCNH2HTR1ATMEM97
Trifluoroacetic Acid SCHEMBL29208064 0.84 HTR2A (0.39) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL30832015 0.82 HTR2A (0.52) HTR2AHTR2CKCNH2HTR1ATMEM97
Trifluoroacetic Acid SCHEMBL29207981 0.81 ALDH1A1 (0.44) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL30832029 0.79 HTR2A (0.42) HTR2AHTR2CKCNH2HTR1ATMEM97
Trifluoroacetic Acid SCHEMBL29207974 0.79 HTR2A (0.48) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL29280918 0.75 GABRA5 (0.47) HTR2AHTR2CKCNH2HTR1ATMEM97
SCHEMBL29208006 0.74 HTR2A (0.54) HTR2AHTR2CKCNH2HTR1ATMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed