SCHEMBL30831998

SCHEMBL30831998

Cc1ccc(CNC(=O)N(C)CC2CCN(CC(=O)c3ccc(F)cc3)CC2)cn1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.42
KCNH2 Q12809 3/20 0.42
KDM4E B2RXH2 3/20 0.42
POLB P06746 1/20 0.42
HTR2A P28223 4/20 0.41
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR2C P28335 2/20 0.40
HTR1A P08908 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
DRD2 P14416 1/20 0.39
HTR2B P41595 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29207960 0.95 HRH3 (0.39) HRH3KCNH2KDM4EPOLBHTR2A
SCHEMBL30832023 0.89 MLLT1 (0.43) HRH3KCNH2KDM4EHTR2AALDH1A1
SCHEMBL30832020 0.88 ALDH1A1 (0.42) HRH3KCNH2KDM4EHTR2AALDH1A1
SCHEMBL30832047 0.87 TSHR (0.47) KDM4EALDH1A1TSHRHTTSMN1; SMN2
SCHEMBL30842099 0.87 HTR2A (0.42) HRH3KCNH2HTR2AHTR2CHTR2B
SCHEMBL30842003 0.86 HRH3 (0.42) HRH3KCNH2HTR2AALDH1A1TSHR
SCHEMBL29208106 0.85 HTR2A (0.51) KCNH2HTR2AHTTSMN1; SMN2HTR2C
SCHEMBL30832022 0.84 ALDH1A1 (0.41) HRH3KCNH2KDM4EHTR2AALDH1A1
SCHEMBL30832039 0.84 ALDH1A1 (0.54) HRH3KCNH2HTR2AALDH1A1TSHR
SCHEMBL30832045 0.83 LMNA (0.52) HRH3KDM4EHTR2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed