SCHEMBL30832008

SCHEMBL30832008

COCc1ccc(NC(=O)N(C)CC2CCN(CC(=O)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 2/20 0.44
HTT P42858 1/20 0.44
MAPT P10636 1/20 0.44
CCR3 P51677 1/20 0.42
TP53 P04637 1/20 0.41
HTR2A P28223 3/20 0.41
HTR2C P28335 2/20 0.41
KCNH2 Q12809 1/20 0.41
HTR1A P08908 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
DRD2 P14416 1/20 0.40
HTR2B P41595 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29207949 0.95 SMN1; SMN2 (0.41) ALDH1A1SMN1; SMN2LMNAHTTMAPT
SCHEMBL30832012 0.89 HTR2A (0.46) SMN1; SMN2LMNAHTR2AHTR2CKCNH2
SCHEMBL30842115 0.87 CYP2D6 (0.41) ALDH1A1SMN1; SMN2LMNAHTTMAPT
SCHEMBL30842106 0.87 DEGS1 (0.40) ALDH1A1SMN1; SMN2HTTHTR2AHTR2C
SCHEMBL30832024 0.86 HTR2A (0.41) HTR2AHTR2CKCNH2HTR1ATMEM97
Trifluoroacetic Acid SCHEMBL29208051 0.84 HTR2A (0.42) HTR2AHTR2CKCNH2
SCHEMBL30832017 0.83 SMN1; SMN2 (0.42) ALDH1A1SMN1; SMN2LMNAHTTMAPT
Trifluoroacetic Acid SCHEMBL29207977 0.83 CYP2D6 (0.38) ALDH1A1SMN1; SMN2LMNAHTTMAPT
Trifluoroacetic Acid SCHEMBL29208058 0.83 HTR2A (0.37) ALDH1A1SMN1; SMN2HTTHTR2AHTR2C
SCHEMBL30831994 0.82 KMT2A (0.42) ALDH1A1HTR2AHTR2CKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed