SCHEMBL30832012

SCHEMBL30832012

COCc1ccc(CNC(=O)N(C)CC2CCN(CC(=O)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.46
HRH3 Q9Y5N1 3/20 0.46
KMT2A Q03164 1/20 0.43
KCNH2 Q12809 2/20 0.42
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTR2C P28335 1/20 0.41
HTR1A P08908 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29208051 0.95 HTR2A (0.42) HTR2AHRH3KMT2AKCNH2HTR2C
SCHEMBL30832045 0.91 LMNA (0.52) HTR2AHRH3KMT2ALMNATSHR
SCHEMBL29207983 0.90 HTR2A (0.49) HTR2AHRH3KMT2AKCNH2HTR2C
SCHEMBL30832008 0.89 ALDH1A1 (0.44) HTR2AKCNH2LMNASMN1; SMN2HTR2C
SCHEMBL30842023 0.89 HTR2A (0.41) HTR2AHRH3KCNH2HTR2C
SCHEMBL30842099 0.89 HTR2A (0.42) HTR2AHRH3KCNH2HTR2C
SCHEMBL29208106 0.88 HTR2A (0.51) HTR2AKMT2AKCNH2SMN1; SMN2HTR2C
SCHEMBL30832034 0.88 HRH3 (0.51) HTR2AHRH3KCNH2LMNATSHR
SCHEMBL30832039 0.87 ALDH1A1 (0.54) HTR2AHRH3KMT2AKCNH2TSHR
SCHEMBL29208114 0.87 HTR2A (0.43) HTR2AHRH3KMT2AKCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed