SCHEMBL30832017

SCHEMBL30832017

COc1ccc(NC(=O)N(C)CC2CCN(CC(=O)c3ccc(F)cc3)CC2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.42
LMNA P02545 3/20 0.42
RAB9A P51151 2/20 0.42
CXCR1 P25024 2/20 0.42
CXCR2 P25025 2/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 4/20 0.41
MAPT P10636 2/20 0.41
HTT P42858 2/20 0.41
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TSHR P16473 1/20 0.40
GALR3 O60755 1/20 0.40
HTR2A P28223 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR1A P08908 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29207991 0.95 PRKAB2 (0.40) SMN1; SMN2LMNARAB9ACXCR1CXCR2
SCHEMBL30842115 0.88 CYP2D6 (0.41) SMN1; SMN2LMNAALDH1A1MAPTHTT
SCHEMBL30832023 0.87 MLLT1 (0.43) SMN1; SMN2LMNAALDH1A1HTTKDM4E
SCHEMBL30831999 0.84 ALDH1A1 (0.43) SMN1; SMN2LMNAALDH1A1HTTKDM4E
SCHEMBL30832008 0.83 ALDH1A1 (0.44) SMN1; SMN2LMNAALDH1A1MAPTHTT
Trifluoroacetic Acid SCHEMBL29207977 0.83 CYP2D6 (0.38) SMN1; SMN2LMNAALDH1A1MAPTHTT
Trifluoroacetic Acid SCHEMBL29207943 0.83 MLLT1 (0.40) HTR2AHTR2CKCNH2
SCHEMBL30832010 0.81 MEN1 (0.41) SMN1; SMN2ALDH1A1HTTKDM4EMEN1
SCHEMBL30842106 0.80 DEGS1 (0.40) SMN1; SMN2ALDH1A1HTTKDM4ETSHR
SCHEMBL29220441 0.78 HTR2A (0.45) SMN1; SMN2LMNARAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed