SCHEMBL30833450

SCHEMBL30833450

CC(F)(C1CCN(C(=O)Nc2ccno2)CC1)S(=O)(=O)c1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
CACNA1B Q00975 3/20 0.45
NR1I2 O75469 2/20 0.45
TSHR P16473 1/20 0.42
NPC1 O15118 1/20 0.41
SCD5 Q86SK9 1/20 0.38
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.38
HPGDS O60760 1/20 0.37
ALDH1A1 P00352 2/20 0.37
USP2 O75604 2/20 0.37
CYP2C9 P11712 2/20 0.37
HIF1A Q16665 1/20 0.37
CYP1A2 P05177 1/20 0.36
SPR P35270 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17942403 1.00 CYP3A4 (0.45) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL17948943 0.84 TSHR (0.47) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL29530688 0.84 TSHR (0.47) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL30833388 0.83 RIPK1 (0.38) CYP3A4CACNA1BNR1I2SCD5KMT2A
SCHEMBL17949487 0.83 FAAH (0.50) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL17949198 0.83 TSHR (0.48) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL17948950 0.83 NPC1 (0.47) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL17949199 0.83 TSHR (0.48) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL17949176 0.83 NR1I2 (0.44) CYP3A4CACNA1BNR1I2TSHRNPC1
SCHEMBL17948942 0.83 NR1I2 (0.44) CYP3A4CACNA1BNR1I2TSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118164961-A 4-Methylsulfonyl substituted piperidine urea compounds for the treatment of Dilated Cardiomyopathy (DCM) 迈奥卡迪亚公司 2024-06-11 CN disclosed
CN-111393414-B 4-Methylsulfonyl substituted piperidine urea compounds for the treatment of Dilated Cardiomyopathy (DCM) 迈奥卡迪亚公司 2024-05-07 CN disclosed