SCHEMBL30833709

SCHEMBL30833709

O=[SH](=O)NCc1ccccc1Nc1nc(Nc2ccc3c(c2)OCO3)ncc1Br

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.55
IGF1R P08069 4/20 0.50
STK17B O94768 1/20 0.45
STK17A Q9UEE5 1/20 0.45
MAPK8 P45983 2/20 0.44
ULK1 O75385 5/20 0.43
CHEK1 O14757 1/20 0.43
FLT3 P36888 1/20 0.43
BRD4 O60885 2/20 0.41
CLK1 P49759 1/20 0.41
CLK2 P49760 1/20 0.41
DYRK1A Q13627 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
GSK3B P49841 1/20 0.41
CDK19 Q9BWU1 1/20 0.41
ALK Q9UM73 1/20 0.41
SYK P43405 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833779 0.84 EGFR (0.48) CDK1IGF1RMAPK8ULK1GSK3B
SCHEMBL29190667 0.81 CDK1 (0.56) CDK1IGF1RSTK17BSTK17AMAPK8
SCHEMBL29190630 0.80 EGFR (0.54) CDK1IGF1RSTK17AMAPK8ULK1
SCHEMBL30833768 0.79 ALK (0.46) CDK1IGF1RSTK17AMAPK8CLK2
SCHEMBL21374195 0.79 CDK1 (0.56) CDK1IGF1RSTK17AMAPK8ULK1
SCHEMBL30833671 0.79 JAK2 (0.42) CDK1IGF1RSTK17AMAPK8ULK1
SCHEMBL30833634 0.79 IGF1R (0.46) IGF1RMAPK8
SCHEMBL29190628 0.79 IGF1R (0.46) IGF1RMAPK8
SCHEMBL30833790 0.79 IGF1R (0.44) CDK1IGF1RMAPK8CDK19ALK
SCHEMBL30833758 0.78 SYK (0.46) IGF1RSTK17AMAPK8CLK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed