SCHEMBL30833713

SCHEMBL30833713

CN1CCN(c2cnc3cc(Nc4ncc(Cl)c(Nc5ccccc5CS(N)(=O)=O)n4)ccc3n2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 4/20 0.52
MAP3K7 O43318 3/20 0.52
NEK2 P51955 1/20 0.52
CCNK O75909 2/20 0.51
CCNA2 P20248 2/20 0.51
CDK2 P24941 2/20 0.51
CCND3 P30281 2/20 0.51
CDK9 P50750 2/20 0.51
CDK6 Q00534 2/20 0.51
ALK Q9UM73 4/20 0.51
FLT3 P36888 1/20 0.51
EGFR P00533 2/20 0.49
SLC2A1 P11166 1/20 0.49
BRD4 O60885 4/20 0.48
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
FGFR1 P11362 1/20 0.48
SRC P12931 1/20 0.48
MAPK1 P28482 1/20 0.48
MAP2K1 Q02750 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833720 0.97 AXL (0.52) AXLMAP3K7NEK2CCNKCCNA2
SCHEMBL30833668 0.91 EGFR (0.52) ALKFLT3EGFRBRD4FGFR1
SCHEMBL30833637 0.86 MAP3K7 (0.53) AXLMAP3K7NEK2CCNKCCNA2
SCHEMBL29190637 0.86 ALK (0.65) AXLMAP3K7NEK2CCNKCCNA2
SCHEMBL30833800 0.83 MAP3K7 (0.53) AXLMAP3K7NEK2CCNKCCNA2
SCHEMBL29190531 0.83 ALK (0.65) AXLMAP3K7NEK2CCNKCCNA2
SCHEMBL30833714 0.77 ALK (0.46) AXLNEK2CDK2CDK9ALK
SCHEMBL30833735 0.77 EGFR (0.52) MAP3K7FLT3EGFRFGFR1SRC
SCHEMBL29190583 0.76 EGFR (0.59) ALKFLT3EGFRBRD4ROS1
SCHEMBL30833776 0.76 ALK (0.48) ALKFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed