SCHEMBL30833750

SCHEMBL30833750

CC(C)(C)OC(=O)N(C(=O)OC(C)(C)C)c1nn(C(=O)OC(C)(C)C)c2cc(N)ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 1/20 0.39
NR1H2 P55055 1/20 0.39
KDR P35968 2/20 0.33
BRD4 O60885 2/20 0.33
RET P07949 1/20 0.33
PDGFRA P16234 1/20 0.32
CDK5 Q00535 1/20 0.32
TYRO3 Q06418 1/20 0.32
SMARCA2 P51531 1/20 0.31
SMARCA4 P51532 1/20 0.31
PBRM1 Q86U86 1/20 0.31
F12 P00748 3/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
PIK3CD O00329 1/20 0.31
ABL1 P00519 1/20 0.31
EGFR P00533 1/20 0.31
HCK P08631 1/20 0.31
SRC P12931 1/20 0.31
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190565 0.91 NR1H2 (0.34) MAP2K4NR1H2BRD4PDGFRACDK5
SCHEMBL1316854 0.86 PDGFRA (0.42) MAP2K4PDGFRACDK5TYRO3PDPK1
SCHEMBL1321196 0.83 MAP2K4 (0.39) MAP2K4
SCHEMBL23559619 0.83 MAP2K4 (0.37) MAP2K4BRD4RET
SCHEMBL29139296 0.83 MAP2K4 (0.43) MAP2K4NR1H2BRD4RORC
Potassium Ion SCHEMBL1317651 0.82 MAP2K4 (0.39) MAP2K4
SCHEMBL30833809 0.82 ELANE (0.41) MAP2K4BRD4GABRG2GABRB3GABRA5
SCHEMBL426350 0.81 NR1H2 (0.42) MAP2K4NR1H2KDRBRD4RET
SCHEMBL3516297 0.81 ELANE (0.35) MAP2K4NR1H2BRD4PDPK1CHEK1
SCHEMBL6168961 0.80 NR1H2 (0.41) MAP2K4NR1H2KDRBRD4RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed