SCHEMBL30833762

SCHEMBL30833762

Nc1ccc2c(N3CCC(N4CCOCC4)CC3)n[nH]c2c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.44
HRH3 Q9Y5N1 6/20 0.43
PDPK1 O15530 1/20 0.39
JAK2 O60674 1/20 0.38
PIK3CA P42336 1/20 0.38
AXL P30530 1/20 0.38
FGFR1 P11362 2/20 0.37
FLT1 P17948 1/20 0.37
KDR P35968 1/20 0.37
MAP4K4 O95819 1/20 0.36
L3MBTL3 Q96JM7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
KCNH2 Q12809 2/20 0.36
CHIT1 Q13231 1/20 0.36
DDR2 Q16832 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190689 1.00 MAPK1 (0.44) MAPK1HRH3PDPK1JAK2PIK3CA
SCHEMBL29190556 0.87 MAPK1 (0.54) MAPK1PDPK1JAK2PIK3CAAXL
SCHEMBL29190522 0.86 KCNH2 (0.44) MAPK1JAK2AXLFGFR1FLT1
SCHEMBL30833743 0.86 KCNH2 (0.44) MAPK1JAK2AXLFGFR1FLT1
SCHEMBL30833680 0.81 MAPK1 (0.43) MAPK1HRH3L3MBTL1
SCHEMBL29190586 0.81 MAPK1 (0.43) MAPK1HRH3L3MBTL1
SCHEMBL30833677 0.81 MAPK1 (0.43) MAPK1HRH3L3MBTL1
SCHEMBL761105 0.77 MAPK1 (0.54) MAPK1PDPK1JAK2PIK3CAAXL
SCHEMBL30833725 0.74 AXL (0.50) MAPK1JAK2AXL
SCHEMBL4785556 0.74 AXL (0.50) MAPK1JAK2AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed