SCHEMBL30843259

SCHEMBL30843259

COc1ccc2cc(Cn3ncc4c(Cl)ccc(C(=O)O)c43)ccc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 2/20 0.39
EGLN1 Q9GZT9 1/20 0.38
P2RX3 P56373 2/20 0.38
PDE5A O76074 1/20 0.38
TDP1 Q9NUW8 2/20 0.37
POLB P06746 1/20 0.37
CCR2 P41597 3/20 0.36
PPARG P37231 1/20 0.36
KLKB1 P03952 3/20 0.35
KLK1 P06870 2/20 0.35
PRKAG1 P54619 2/20 0.35
PRKAA1 Q13131 2/20 0.35
PRKAB1 Q9Y478 2/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
PTGER4 P35408 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21458280 1.00 NPBWR1 (0.39) NPBWR1EGLN1P2RX3PDE5ATDP1
SCHEMBL30843280 0.91 NPBWR1 (0.39) NPBWR1EGLN1P2RX3TDP1KLKB1
SCHEMBL21458219 0.91 NPBWR1 (0.39) NPBWR1EGLN1P2RX3TDP1KLKB1
SCHEMBL24992167 0.82 CRHR1 (0.39) PDE5A
SCHEMBL30843267 0.82 PTGER4 (0.40) P2RX3KLKB1KLK1PTGER4
SCHEMBL21458242 0.82 PTGER4 (0.40) P2RX3KLKB1KLK1PTGER4
SCHEMBL21481962 0.80 CHRM4 (0.35) KLKB1KLK1PTGER4
SCHEMBL21458140 0.80 CHRM4 (0.35) KLKB1KLK1PTGER4
SCHEMBL21481961 0.77 CNR2 (0.40) PDE5AMTNR1AMTNR1B
SCHEMBL21481971 0.77 CRHR1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250353829-A1 BICYCLIC CARBOXAMIDES AND METHODS OF USE THEREOF TEMPEST THERAPEUTICS INC (US) 2025-11-20 US disclosed
CN-112313208-B Bicyclic carboxamides and methods of use thereof 泰普斯特医疗公司 2024-04-19 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250353829-A1 BICYCLIC CARBOXAMIDES AND METHODS OF USE THEREOF PTGER4, PTGER2, CNR2 NPBWR1 635/4885EGLN1 336/4885P2RX3 70/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.