SCHEMBL30845404

SCHEMBL30845404

COC(=O)c1csc2cccnc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 5/20 0.55
KDM4E B2RXH2 4/20 0.52
MAP2K1 Q02750 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
CHEK1 O14757 1/20 0.46
MET P08581 1/20 0.46
GSK3B P49841 1/20 0.46
LIMK1 P53667 1/20 0.46
DYRK1A Q13627 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
DYRK1B Q9Y463 1/20 0.46
PSMD14 O00487 1/20 0.43
ALDH1A1 P00352 1/20 0.43
SLC40A1 Q9NP59 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
IRAK1 P51617 1/20 0.42
SYK P43405 2/20 0.42
AURKA O14965 1/20 0.42
MAP3K7 O43318 1/20 0.42
FLT3 P36888 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29560146 0.84 IRAK4 (0.46) IRAK4KDM4ELIMK1ALDH1A1IRAK1
SCHEMBL17023631 0.82 IRAK4 (0.49) IRAK4KDM4ELIMK1ALDH1A1L3MBTL1
SCHEMBL29560247 0.80 KDM4E (0.48) IRAK4KDM4ETDP1LIMK1ALDH1A1
SCHEMBL7114666 0.80 KDM4E (0.48) IRAK4KDM4ETDP1LIMK1ALDH1A1
SCHEMBL30844941 0.79 PARP1 (0.53) IRAK4KDM4ELIMK1ALDH1A1L3MBTL1
SCHEMBL19555042 0.79 PARP1 (0.53) IRAK4KDM4ELIMK1ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL30845090 0.78 PARP1 (0.51) IRAK4KDM4ELIMK1ALDH1A1L3MBTL1
SCHEMBL29559995 0.77 IRAK4 (0.51) IRAK4ALDH1A1IRAK1SYKAURKA
SCHEMBL15466759 0.76 ALDH1A1 (0.46) KDM4ETDP1PSMD14ALDH1A1POLB
Water SCHEMBL30682486 0.76 IRAK4 (0.50) IRAK4ALDH1A1IRAK1SYKAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113423711-B Thieno [3,2-B ] pyridine derivatives as UDP glycosyltransferase inhibitors and methods of use thereof 建新公司 2024-03-15 CN disclosed