SCHEMBL30844941

SCHEMBL30844941

NC(=O)c1csc2cccnc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.53
LIMK1 P53667 2/20 0.51
KDM4E B2RXH2 3/20 0.49
IRAK4 Q9NWZ3 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.41
PLK4 O00444 1/20 0.40
MAP4K4 O95819 1/20 0.40
EGFR P00533 1/20 0.40
ROS1 P08922 1/20 0.40
PIM1 P11309 1/20 0.40
AXL P30530 1/20 0.40
FLT3 P36888 1/20 0.40
FRK P42685 1/20 0.40
MAP4K2 Q12851 1/20 0.40
NTRK3 Q16288 1/20 0.40
MINK1 Q8N4C8 1/20 0.40
AURKB Q96GD4 1/20 0.40
HIPK2 Q9H2X6 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
STK17A Q9UEE5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19555042 1.00 PARP1 (0.53) PARP1LIMK1KDM4EIRAK4L3MBTL1
Hydrochloric Acid SCHEMBL30845090 0.98 PARP1 (0.51) PARP1LIMK1KDM4EIRAK4L3MBTL1
Trifluoroacetic Acid SCHEMBL30844916 0.90 L3MBTL1 (0.50) PARP1LIMK1KDM4EIRAK4L3MBTL1
SCHEMBL7114666 0.84 KDM4E (0.48) LIMK1KDM4EIRAK4L3MBTL1IRAK1
SCHEMBL29560247 0.84 KDM4E (0.48) LIMK1KDM4EIRAK4L3MBTL1IRAK1
SCHEMBL17023631 0.83 IRAK4 (0.49) PARP1LIMK1KDM4EIRAK4L3MBTL1
SCHEMBL8555310 0.82 IRAK4 (0.44) PARP1LIMK1KDM4EIRAK4L3MBTL1
SCHEMBL30845404 0.79 IRAK4 (0.55) LIMK1KDM4EIRAK4L3MBTL1FLT3
SCHEMBL3385296 0.76 LIMK1 (0.44) PARP1LIMK1KDM4EIRAK4L3MBTL1
SCHEMBL29560146 0.75 IRAK4 (0.46) LIMK1KDM4EIRAK4FLT3IRAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113423711-B Thieno [3,2-B ] pyridine derivatives as UDP glycosyltransferase inhibitors and methods of use thereof 建新公司 2024-03-15 CN claimed
CN-118239963-A Compounds as eIF4E inhibitors and uses thereof 南京圣和药业股份有限公司 2024-06-25 CN disclosed
CN-113423711-B Thieno [3,2-B ] pyridine derivatives as UDP glycosyltransferase inhibitors and methods of use thereof 建新公司 2024-03-15 CN disclosed